2/11/2004
FARM 2147 Fluoroquinolones
23
1960
1970
1980
1990
2000
• Temafloxacin a
• Sparfloxacin b
• Grepafloxacin c
•  Gatifloxacin d
 The “second generation” fluoroquinolones
• Gram (-);
  • improved
  Gram (+)
anti-anaerobe
a: Toyama, 1988 (?) ; b: Dainippon, 1985-1987; c: Otskuda, 1989; d: Kyorin, 1988