TARGETS FOR DRUG ACTION
Transporters
Carriers
Inhibitors
False
substrates
Choline carrier
(nerve terminal)
Hemicholinium
Noradrenaline
uptake1
Tricyclic
antidepressants
Cocaine
Amphetamine
Methyldopa
Noradrenaline
uptake (vesicular)
Reserpine
Weak acid carrier
(renal tubule)
Probenecid
Na+/K+/Cl- co-
transporter (loop
of Henle)
Loop diuretics
Na+/K+ pump
Cardiac
glycosides
Proton pump
(gastric mucosa)
Omeprazole
2003-2004