TARGETS FOR DRUG ACTION
Receptors
Danazol
Norethisterone
Progesterone
receptor
Tamoxifen
Ethinylestradiol
Oestrogen
receptor
Not known
Insulin
Insulin receptor
Chlorpromazine
Dopamine
Bromocriptine
Dopamine (D2-
receptor)
Ketanserine
5-
hydroxytryptamine
5HT2 receptor
Naloxone
Morphine
Opiate (
µ
- )
receptor)
Ranitidine
Impromidine
Histamine (H2 -
receptor)
Mepyramine
Histamine
Histamine (H1-
receptor
Propranolol
Noradrenaline
Isoprenaline
Beta-adreno-
receptor
Tubocurarine
a
-bungarotoxin
Acetylcholine
Nicotine
Nicotinic Ach
receptor
Antagonists
Agonists
Receptors
From Pharmacology
Ed Rang et al (2003)
Churchill Livingstone, p 23
2003-2004