2/11/2004
FARM 2147 Fluoroquinolones
1960
1970
1980
1990
2000
• Temafloxacin a
• Sparfloxacin b
• Grepafloxacin c
• Gatifloxacin d
The “second generation” fluoroquinolones
• Gram
(-);
• improved
Gram (+)
anti-anaerobe
a: Toyama,
1988 (?) ; b: Dainippon, 1985-1987; c: Otskuda, 1989; d: Kyorin, 1988