2/11/2004
FARM 2147 Fluoroquinolones
Ternary
complex
DNA - enzyme -
fluoroquinolone
FLUOROQUINOLONES:
4 stacked molecules
DNA GYRASE
catalytic subunits
DNA GYRASE
ATP binding subunits
COVALENTLY CLOSED
CIRCULAR DNA
(Shen, in Quinolone Antimicrobial Agents, 1993)